Identification of inhibitors of Tartrate-resistant acid phosphatase (TRAP/ACP5 ) activity by small-molecule screening-Reference-Cited by-同舟云学术

Identification of inhibitors of Tartrate-resistant acid phosphatase (TRAP/ACP5 ) activity by small-molecule screening

Published:2018-03-30 Issue:1 Volume:92 Page:1255-1271
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Reithmeier Anja¹^ORCID,Lundbäck Thomas²,Haraldsson Martin²,Frank Martin³,Ek-Rylander Barbro¹,Nyholm Per-Georg³,Gustavsson Anna-Lena²,Andersson Göran¹

Affiliation:

1. Department of Laboratory Medicine (LABMED); H5, Division of Pathology, F46; Karolinska University Hospital; Huddinge, Stockholm Sweden

2. Chemical Biology Consortium Sweden (CBCS); Science for Life Laboratory; Department of Medical Biochemistry and Biophysics; Karolinska Institutet; Stockholm Sweden

3. Biognos AB; Gothenburg Sweden

Funder

Science for Life Laboratories

Cancerfonden

Vetenskapsrådet

Karolinska Institutet

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.13187/fullpdf

Reference56 articles.

1. Structure, function, and regulation of tartrate-resistant acid phosphatase

2. Tartrate-resistant purple acid phosphatase is synthesized as a latent proenzyme and activated by cysteine proteinases

3. Three-dimensional structure of a mammalian purple acid phosphatase at 2.2 Å resolution with a μ-(hydr)oxo bridged di-iron center

4. Crystal structure of a mammalian purple acid phosphatase 1 1Edited by R. Huber

5. Crystal structure of mammalian purple acid phosphatase

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