Profiling two indole-2-carboxamides for allosteric modulation of the CB1 receptor-Reference-Cited by-同舟云学术

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Profiling two indole-2-carboxamides for allosteric modulation of the CB1 receptor

Published:2013-01-07 Issue:5 Volume:124 Page:584-589
ISSN:0022-3042
Container-title:Journal of Neurochemistry
language:en
Short-container-title:J. Neurochem.

Author:

Ahn Kwang H.¹,Mahmoud Mariam M.²,Samala Sushma³,Lu Dai³,Kendall Debra A.¹

Affiliation:

1. Department of Pharmaceutical Sciences; University of Connecticut; Storrs Connecticut USA

2. Department of Molecular and Cell Biology; University of Connecticut; Storrs Connecticut USA

3. Department of Pharmaceutical Sciences; Irma Lerma Rangel College of Pharmacy; Texas A&M Health Science Center; Kingsville Texas USA

Funder

National Institutes of Health Grant

Texas A&M Health Sciences Center

Publisher

Wiley

Subject

Cellular and Molecular Neuroscience,Biochemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/jnc.12115/fullpdf

Reference13 articles.

1. Desensitization, internalization, and signaling functions of beta-arrestins demonstrated by RNA interference;Ahn;Proc. Natl Acad. Sci. USA,2003

2. Dual role of the second extracellular loop of the cannabinoid receptor 1: ligand binding and receptor localization;Ahn;Mol. Pharmacol.,2009

3. Allosteric modulator ORG27569 induces CB1 cannabinoid receptor high affinity agonist binding state, receptor internalization, and Gi protein-independent ERK1/2 kinase activation;Ahn;J. Biol. Chem.,2012

4. High-efficiency transformation of mammalian cells by plasmid DNA;Chen;Mol. Cell. Biol.,1987

5. Cannabinoid transmission and reward-related events;Gardner;Neurobiol. Dis.,1998

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1. Membrane Lipids Are an Integral Part of Transmembrane Allosteric Sites in GPCRs: A Case Study of Cannabinoid CB1 Receptor Bound to a Negative Allosteric Modulator, ORG27569, and Analogs;Journal of Medicinal Chemistry;2022-09-06

2. The type 1 cannabinoid receptor positive allosteric modulators GAT591 and GAT593 reduce spike-and-wave discharges in Genetic Absence Epilepsy Rats from Strasbourg;IBRO Neuroscience Reports;2022-06

3. Rational design of cannabinoid type-1 receptor allosteric modulators: Org27569 and PSNCBAM-1 hybrids;Bioorganic & Medicinal Chemistry;2021-07

4. CB1 allosteric modulators and their therapeutic potential in CNS disorders;Progress in Neuro-Psychopharmacology and Biological Psychiatry;2021-03

5. Protein Interactors and Trafficking Pathways That Regulate the Cannabinoid Type 1 Receptor (CB1R);Frontiers in Molecular Neuroscience;2020-06-12

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