Structure-Based Grafting, Mutation, and Optimization of Peptide Inhibitors to Fit in the Active Pocket of Human Secreted Phospholipase A2: Find New Use of Old Peptide Agents with Anti-Inflammatory Activity-Reference-Cited by-同舟云学术

Structure-Based Grafting, Mutation, and Optimization of Peptide Inhibitors to Fit in the Active Pocket of Human Secreted Phospholipase A2: Find New Use of Old Peptide Agents with Anti-Inflammatory Activity

Published:2014-09-25 Issue:4 Volume:85 Page:418-426
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Zhan Chengye¹,Li Shusheng¹,Zhong Qiang¹,Zhou Daixing¹

Affiliation:

1. Department of ICU; Tongji Hospital; Tongji Medical College; Huazhong University of Science and Technology; Wuhan 430030 China

Funder

Foundation of Science Technology Department of Hubei Province, China

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.12424/fullpdf

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3. Secretory non-pancreatic group II phospholipase A2: role in physiologic and inflammatory processes;Pruzanski;J Lipid Mediat,1993

4. Recombinant secreted nonpancreatic phospholipase A2 induces a synovitis-like inflammation in the rat air pouch;Cirino;J Rheumatol,1994

5. Secretory phospholipases A2 induce cytokine release from blood and synovial fluid monocytes;Triggiani;Eur J Immunol,2002

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