A novel fluorophosphonate inhibitor of the biosynthesis of the endocannabinoid 2-arachidonoylglycerol with potential anti-obesity effects

Author:

Bisogno Tiziana,Mahadevan Anu1,Coccurello Roberto2,Chang Jae Won3,Allarà Marco4,Chen Yugang1,Giacovazzo Giacomo2,Lichtman Aron5,Cravatt Benjamin3,Moles Anna,Di Marzo Vincenzo4

Affiliation:

1. Organix Inc.; Woburn; MA; USA

2. Cell Biology and Neurobiology Institute (IBCN)/IRCCS Fondazione Santa Lucia; Roma; Italy

3. The Skaggs Institute for Chemical Biology and Department of Chemical Physiology; The Scripps Research Institute; La Jolla; CA; USA

4. Endocannabinoid Research Group; Institute of Biomolecular Chemistry; C.N.R.; Pozzuoli; Italy

5. Department of Pharmacology and Toxicology; Virginia Commonwealth University; Richmond; VA; USA

Publisher

Wiley

Subject

Pharmacology

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