Pharmacokinetics and tolerability of eslicarbazepine acetate and oxcarbazepine at steady state in healthy volunteers

Author:

Elger Christian1,Bialer Meir2,Falcão Amílcar3,Vaz-da-Silva Manuel45,Nunes Teresa4,Almeida Luís6,Soares-da-Silva Patrício45

Affiliation:

1. Department of Epileptology; University of Bonn; Bonn Germany

2. Institute for Drug Research; Faculty of Medicine; School of Pharmacy; Hebrew University of Jerusalem; Jerusalem Israel

3. Faculty of Pharmacy; University of Coimbra; Coimbra Portugal

4. BIAL - Portela & Cª, S.A.; S. Mamede do Coronado Portugal

5. Faculty of Medicine; University of Porto; Porto Portugal

6. Health Sciences Department; University of Aveiro; Aveiro Portugal

Funder

BIAL - Portela & Cª, S.A.

Publisher

Wiley

Subject

Clinical Neurology,Neurology

Reference36 articles.

1. Effects of eslicarbazepine, R-licarbazepine and oxcarbazepine on fast and slow inactivation of voltage-gated sodium channels;Aires;Epilepsia,2012

2. Safety, tolerability, and pharmacokinetic profile of BIA 2-093, a novel putative antiepileptic, in a rising multiple-dose study in young healthy humans;Almeida;J Clin Pharmacol,2004

3. Eslicarbazepine acetate (BIA 2-093);Almeida;Neurotherapeutics,2007

4. Single-dose and steady-state pharmacokinetics of eslicarbazepine acetate (BIA 2-093) in healthy elderly and young subjects;Almeida;J Clin Pharmacol,2005

5. Pharmacokinetics, efficacy, and tolerability of eslicarbazepine acetate in children and adolescents with epilepsy;Almeida;J Clin Pharmacol,2008a

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