Pharmacokinetic interaction between the CYP3A4 inhibitor ketoconazole and the hormone drospirenone in combination with ethinylestradiol or estradiol-Reference-Cited by-同舟云学术

Pharmacokinetic interaction between the CYP3A4 inhibitor ketoconazole and the hormone drospirenone in combination with ethinylestradiol or estradiol

Published:2015-10-28 Issue:6 Volume:80 Page:1399-1410
ISSN:0306-5251
Container-title:British Journal of Clinical Pharmacology
language:en
Short-container-title:Br J Clin Pharmacol

Author:

Wiesinger Herbert¹,Berse Matthias²,Klein Stefan¹,Gschwend Simone¹,Höchel Joachim¹,Zollmann Frank S.³,Schütt Barbara¹

Affiliation:

1. Bayer Pharma AG; Berlin

2. CRS Clinical Research Services Berlin GmbH; Berlin

3. Pharma Consult; Berlin Germany

Publisher

Wiley

Subject

Pharmacology (medical),Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/bcp.12745/fullpdf

Reference30 articles.

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2. Bayer Summary of product characteristics: YAZ 0.02 mg/3 mg film coated tablets. 2015 http://www.medicines.ie/medicine/13973/SPC/Yaz+0.02mg+++3mg+film+coated+tablets

3. US Food and Drug Administration Center for Drug Evaluation and Research: NDA 202-258 - Secondary clinical pharmacology review 2011 http://www.accessdata.fda.gov/drugsatfda_docs/nda/2011/202258orig1s000clinpharmr.pdf

4. General framework for the quantitative prediction of CYP3A4-mediated oral drug interactions based on the AUC increase by coadministration of standard drugs;Ohno;Clin Pharmacokinet,2007

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