Design, synthesis, and biologic evaluation of novel galloyl derivatives as HIV ‐1 RN ase H inhibitors-Reference-Cited by-同舟云学术

Design, synthesis, and biologic evaluation of novel galloyl derivatives as HIV ‐1 RN ase H inhibitors

Published:2019-01-24 Issue:4 Volume:93 Page:582-589
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Gao Ping¹,Wang Xueshun¹,Sun Lin¹,Cheng Xiqiang¹,Poongavanam Vasanthanathan²,Kongsted Jacob²,Álvarez Mar³,Luczkowiak Joanna³,Pannecouque Christophe⁴,De Clercq Erik⁴,Lee Kuo‐Hsiung⁵,Chen Chin‐Ho⁶,Liu Huiqing⁷,Menéndez‐Arias Luis³^ORCID,Liu Xinyong¹^ORCID,Zhan Peng¹^ORCID

Affiliation:

1. Department of Medicinal ChemistryKey Laboratory of Chemical BiologyMinistry of EducationSchool of Pharmaceutical SciencesShandong University Ji'nan China

2. Department of Physics, Chemistry and PharmacyUniversity of Southern Denmark Odense M Denmark

3. Centro de Biología Molecular “Severo Ochoa” (Consejo Superior de Investigaciones Científicas and Universidad Autónoma de Madrid) Madrid Spain

4. Rega Institute for Medical ResearchK.U.Leuven Leuven Belgium

5. Natural Products Research LaboratoriesEshelman School of PharmacyUniversity of North Carolina Chapel Hill North Carolina

6. Surgical ScienceDepartment of SurgeryDuke University Medical Center Durham North Carolina

7. Department of PharmacologySchool of Basic Medical SciencesShandong University Jinan China

Funder

National Natural Science Foundation of China

Division of Intramural Research, National Institute of Allergy and Infectious Diseases

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1111/cbdd.13455

Reference32 articles.

1. Increased Thermostability and Fidelity of DNA Synthesis of Wild-Type and Mutant HIV-1 Group O Reverse Transcriptases

2. Inhibition of the Ribonuclease H Activity of HIV-1 Reverse Transcriptase by GSK5750 Correlates with Slow Enzyme-Inhibitor Dissociation

3. Design, Synthesis, and Biological Evaluation of a Series of 2-Hydroxyisoquinoline-1,3(2H,4H)-diones as Dual Inhibitors of Human Immunodeficiency Virus Type 1 Integrase and the Reverse Transcriptase RNase H Domain

4. Selective inhibition of HIV-1 reverse transcriptase-associated ribonuclease H activity by hydroxylated tropolones

5. Recent Progress in the Research of Small Molecule HIV-1 RNase H Inhibitors

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