Design, synthesis and antitrypanosomatid activities of 3,5-diaryl-isoxazole analogues based on neolignans veraguensin, grandisin and machilin G-Reference-Cited by-同舟云学术

Design, synthesis and antitrypanosomatid activities of 3,5-diaryl-isoxazole analogues based on neolignans veraguensin, grandisin and machilin G

Published:2018-11-25 Issue:3 Volume:93 Page:313-324
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Trefzger Ozildéia S.¹,das Neves Amarith R.¹²,Barbosa Natália V.¹²,Carvalho Diego B.¹,Pereira Indiara C.³,Perdomo Renata T.³,Matos Maria F. C.³,Yoshida Nidia C.⁴,Kato Massuo J.⁵,de Albuquerque Sérgio⁶,Arruda Carla C. P.²,Baroni Adriano C. M.¹^ORCID

Affiliation:

1. LASQUIM - Laboratório de Síntese e Química Medicinal; FACFAN - Faculdade de Ciências Farmacêuticas, Alimentos e Nutrição; Universidade Federal do Mato Grosso do Sul; UFMS; Campo Grande MS Brazil

2. Laboratorio de Parasitologia Humana; INBIO - Instituto de Biologia; Universidade Federal do Mato Grosso do Sul; Campo Grande MS Brazil

3. Laboratorio de Biologia Molecular e Cultura de Celulas; FACFAN - Faculdade de Ciências Farmacêuticas; Alimentos e Nutricao; Universidade Federal do Mato Grosso do Sul; UFMS; Campo Grande MS Brazil

4. Instituto de Química; Universidade Federal do Mato Grosso do Sul, UFMS; Campo Grande MS Brazil

5. Institute of Chemistry; University of São Paulo; São Paulo SP Brazil

6. Departamento de Análises Clínicas, Toxicológicas e Bromatológicas; Faculdade de Ciências Farmacêuticas de Ribeirão Preto; USP; Ribeirão Preto SP Brazil

Funder

Conselho Nacional de Desenvolvimento Científico e Tecnológico

Fundação de Apoio ao Desenvolvimento do Ensino, Ciência e Tecnologia do Estado de Mato Grosso do Sul

PROPP-UFMS

Coordenação de Aperfeiçoamento de Pessoal de Nível Superior

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.13417/fullpdf

Reference52 articles.

1. Synthesis and trypanocidal activity of 1,4-bis-(3,4,5-trimethoxy-phenyl)-1,4-butanediol and 1,4-bis-(3,4-dimethoxyphenyl)-1,4-butanediol;Bernardes;Bioorganic & Medicinal Chemistry,2006

2. Synthesis and antimalarial activity of quinones and structurally-related oxirane derivatives;Carneiro;European Journal of Medicinal Chemistry,2016

3. Antinociceptive and antiinflammatory activities of grandisin extracted from Virola surinamensis;Carvalho;Phytotherapy Research,2010

4. Synthesis and antitrypanosomastid activity of 1,4-Diaryl-1,2,3-triazole analogues of Neolignans Veraguensin, Grandisin and Machilin G;Cassamale;Journal of the Brazilian Chemical Society,2016

5. A synthetic method for Formyl→ Ethynyl conversion (RCHO → RC≡CH or RC≡CR’);Corey;Tetrahedron Letters,1972

Cited by 24 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Antileishmanial Activity, Toxicity and Mechanism of Action of Complexes of Sodium Usnate with Lanthanide Ions: Eu(III), Sm(III), Gd(III), Nd(III), La(III) and Tb(III);International Journal of Molecular Sciences;2023-12-28

2. Neuroprotective Profile of Triazole Grandisin Analogue against Amyloid-Beta Oligomer-Induced Cognitive Impairment;ACS Chemical Neuroscience;2023-12-04

3. Drug Discovery for Cutaneous Leishmaniasis: A Review of Developments in the Past 15 Years;Microorganisms;2023-11-23

4. Design, synthesis and antitrypanosomatid activity of 2-nitroimidazole-3,5-disubstituted isoxazole compounds based on benznidazole;European Journal of Medicinal Chemistry;2023-11

5. In Vivo Antileishmanial Effect of 3,5-Diaryl-isoxazole Analogues Based on Veraguensin, Grandisin, and Machilin G: A Glance at a Preclinical Study;ACS Infectious Diseases;2023-04-27