First‐in‐human trial to assess the safety, tolerability, pharmacokinetics and pharmacodynamics of STR‐324, a dual enkephalinase inhibitor for pain management-Reference-Cited by-同舟云学术

First‐in‐human trial to assess the safety, tolerability, pharmacokinetics and pharmacodynamics of STR‐324, a dual enkephalinase inhibitor for pain management

Published:2021-07-16 Issue:1 Volume:88 Page:103-114
ISSN:0306-5251
Container-title:British Journal of Clinical Pharmacology
language:en
Short-container-title:Brit J Clinical Pharma

Author:

Moss Laurence M.¹²^ORCID,Berends Cecile L.¹²^ORCID,Brummelen Emilie M. J.¹^ORCID,Kamerling Ingrid M. C.¹²,Klaassen Erica S.¹,Bergmann Kirsten¹,Ville Vanessa³,Juarez‐Perez Victor³,Benichou Annie‐Claude⁴,Groeneveld Geert Jan¹²^ORCID

Affiliation:

1. Centre for Human Drug Research Leiden the Netherlands

2. Leiden University Leiden the Netherlands

3. Stragen France Lyon France

4. Stragen Services Lyon France

Publisher

Wiley

Subject

Pharmacology (medical),Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1111/bcp.14931

Reference26 articles.

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5. Inhibiting the breakdown of endogenous opioids and cannabinoids to alleviate pain

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