Discovery of HIV-1 Integrase Inhibitors: Pharmacophore Mapping, Virtual Screening, Molecular Docking, Synthesis, and Biological Evaluation-Reference-Cited by-同舟云学术

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Discovery of HIV-1 Integrase Inhibitors: Pharmacophore Mapping, Virtual Screening, Molecular Docking, Synthesis, and Biological Evaluation

Published:2013-10-04 Issue:2 Volume:83 Page:154-166
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Bhatt Hardik¹,Patel Paresh²,Pannecouque Christophe³

Affiliation:

1. Department of Pharmaceutical Chemistry; Institute of Pharmacy; Nirma University; Ahmedabad 382 481 India

2. Department of Pharmaceutical Chemistry; L.J. Institute of Pharmacy; L.J. Campus, S.G. Highway Ahmedabad 382 210 India

3. Rega Institute for Medical Research; Minderbroedersstraat 10 B-3000 Leuven Belgium

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.12207/fullpdf

Reference41 articles.

1. Discovery of raltegravir, a potent, selective orally bioavailable HIV-integrase inhibitor for the treatment of HIV-AIDS infection;Summa;J Med Chem,2008

2. New 2-arylnaphthalenediols and triol inhibitors of HIV-1 integrase - Discovery of a new polyhydroxylated antiviral agent;Maurin;Bioorg Med Chem,2010

3. Raltegravir: the First HIV Integrase Inhibitor;Jennifer;Clin Ther,2008

4. Novel quinolinonyl diketo acid derivatives as HIV-1 integrase inhibitors: design, synthesis, and biological activities;Santo;J Med Chem,2008

5. Design and synthesis of novel dihydroquinoline-3-carboxylic acids as HIV-1 integrase inhibitors;Sechi;Bioorg Med Chem,2009

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1. Transition‐Metal Free Arylation of Therapeutically Important Heterocycles;ChemistrySelect;2024-05-15

2. A computational overview of integrase strand transfer inhibitors (INSTIs) against emerging and evolving drug-resistant HIV-1 integrase mutants;Archives of Microbiology;2023-03-26

3. A search for potential anti-HIV phytoconstituents from the natural product repository;Advances in Traditional Medicine;2022-05-14

4. Identification of potent, non-toxic, selective CDK2 inhibitor through the pharmacophore-based scaffold hopping, molecular dynamics simulation-assisted molecular docking study, Lee Richard contour map analysis, and ADMET properties;Structural Chemistry;2022-05-07

5. Bicyclic 6-6 Systems: Pteridines;Comprehensive Heterocyclic Chemistry IV;2022

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