Understanding polyspecificity within the substrate-binding cavity of the human multidrug resistance P-glycoprotein-Reference-Cited by-同舟云学术

Understanding polyspecificity within the substrate-binding cavity of the human multidrug resistance P-glycoprotein

Published:2014-01-17 Issue:3 Volume:281 Page:673-682
ISSN:1742-464X
Container-title:FEBS Journal
language:en
Short-container-title:FEBS J

Author:

Martinez Lorena¹,Arnaud Ophélie¹,Henin Emilie²,Tao Houchao³,Chaptal Vincent¹,Doshi Rupak⁴,Andrieu Thibault⁵,Dussurgey Sébastien⁵,Tod Michel²,Di Pietro Attilio¹,Zhang Qinghai³,Chang Geoffrey⁴,Falson Pierre¹

Affiliation:

1. Drug Resistance Mechanism and Modulation group; Ligue 2013 certified; Molecular and Structural Basis of Infectious Systems; Mixed Research Unit between the National Centre for Scientific Research and Lyon I University n°5086; Institute of Biology and Chemistry of Proteins; France

2. Ciblage Thérapeutique en Oncologie; Mixed Research Team n°3738; Faculté de Médecine Lyon-sud Charles Mérieux; OULLINS Cedex France

3. Department of Integrative Structural and Computational Biology; The Scripps Research Institute; La Jolla CA USA

4. Skaggs School of Pharmacy and Pharmaceutical Sciences; Department of Pharmacology; School of Medicine University of California; San Diego La Jolla CA USA

5. Unité Mixe de Service n°3444; Tour Inserm Cervi; Lyon cedex France

Publisher

Wiley

Subject

Cell Biology,Molecular Biology,Biochemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/febs.12613/fullpdf

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3. The human ATP-binding cassette (ABC) transporter superfamily;Dean;J Lipid Res,2001

4. Targeting multidrug resistance in cancer;Szakacs;Nat Rev Drug Discov,2006

5. ABC efflux pump-based resistance to chemotherapy drugs;Eckford;Chem Rev,2009

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