A partial trace amine-associated receptor 1 agonist exhibits properties consistent with a methamphetamine substitution treatment
Author:
Affiliation:
1. Department of Neuroscience, Psychology and Behaviour; University of Leicester; Leicester UK
2. Neuroscience, Ophthalmology and Rare Diseases Discovery & Translational Area; pRED, Roche Innovation Center Basel; Basel Switzerland
Funder
Hoffmann-La Roche Ltd
Publisher
Wiley
Subject
Psychiatry and Mental health,Pharmacology,Medicine (miscellaneous)
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1111/adb.12410/fullpdf
Reference45 articles.
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2. Mammalian central nervous system trace amines. Pharmacologic amphetamines, physiologic neuromodulators;Berry;J Neurochem,2004
3. Trace amines: identification of a family of mammalian G protein-coupled receptors;Borowsky;Proc Natl Acad Sci,2001
4. The selective antagonist EPPTB reveals TAAR1-mediated regulatory mechanisms in dopaminergic neurons of the mesolimbic system;Bradaia;Proc Natl Acad Sci,2009
5. Amphetamine, 3, 4-methylenedioxymethamphetamine, lysergic acid diethylamide, and metabolites of the catecholamine neurotransmitters are agonists of a rat trace amine receptor;Bunzow;Mol Pharmacol,2001
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