Prolyl hydroxylase inhibition corrects functional iron deficiency and inflammation-induced anaemia in rats

Author:

Barrett Terrance D1,Palomino Heather L2,Brondstetter Theresa I3,Kanelakis Kimon C4,Wu Xiaodong1,Yan Wen5,Merton Katherine P1,Schoetens Freddy1,Ma Jing Ying1,Skaptason Judy1,Gao Jingjin1,Tran Da-Thao1,Venkatesan Hariharan1,Rosen Mark D6,Shankley Nigel P7,Rabinowitz Michael H6

Affiliation:

1. Cardiovascular Metabolic Research; Janssen Pharmaceutical Companies of Johnson & Johnson; San Diego CA USA

2. School of Medicine; University of California at San Diego; San Diego CA USA

3. Covenant Care; Palo Alto CA USA

4. Office of Foods and Veterinary Medicine; U.S. Food and Drug Administration; Rockville MD USA

5. Arcturus Therapeutics; San Diego CA USA

6. Aetheria Therapeutics; San Diego CA USA

7. Higher Todsworthy Farm; Cornwall UK

Funder

Janssen Pharmaceutical Research and Development

Publisher

Wiley

Subject

Pharmacology

Reference28 articles.

1. The Concise Guide to PHARMACOLOGY 2013/14: transporters;Alexander;Br J Pharmacol,2013a

2. The Concise Guide to PHARMACOLOGY 2013/14: enzymes;Alexander;Br J Pharmacol,2013b

3. Pharmacological characterization of 1-(5-chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic acid (JNJ-42041935), a potent and selective hypoxia-inducible factor prolyl hydroxylase inhibitor;Barrett;Mol Pharmacol,2011

4. FG-4592, a novel oral HIF prolyl hydroxylase inhibitor (HIF-PHI), elevates haemoglobin in anemic stage 3-4 CKD patients;Besarab;J Am Soc Nephrol,2010

5. A conserved family of prolyl-4-hydroxylases that modify HIF;Bruick;Science,2001

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