Structures of a diverse set of colchicine binding site inhibitors in complex with tubulin provide a rationale for drug discovery-Reference-Cited by-同舟云学术

Structures of a diverse set of colchicine binding site inhibitors in complex with tubulin provide a rationale for drug discovery

Published:2015-11-04 Issue:1 Volume:283 Page:102-111
ISSN:1742-464X
Container-title:FEBS Journal
language:en
Short-container-title:FEBS J

Author:

Wang Yuxi¹,Zhang Hang¹,Gigant Benoît²,Yu Yamei¹,Wu Yangping¹,Chen Xiangzheng¹,Lai Qinhuai¹,Yang Zhaoya³,Chen Qiang¹,Yang Jinliang¹

Affiliation:

1. State Key Laboratory of Biotherapy and Cancer Center; West China Hospital; Collaborative Innovation Center for Biotherapy; Sichuan University; Chengdu China

2. Institute for Integrative Biology of the Cell (I2BC); CEA; CNRS; Université Paris-Sud; Gif-sur-Yvette France

3. West China School of Pharmacy; Sichuan University; Chengdu China

Funder

National Major Scientific and Technological Special Project

National Natural Science Foundation of China

Scientific Research Foundation for the Returned Overseas Chinese Scholars

Publisher

Wiley

Subject

Cell Biology,Molecular Biology,Biochemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/febs.13555/fullpdf

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4. Alkaloids of Vinca rosea Linn. (Catharanthus roseus G. Don). XV. Analysis of vinca alkaloids by thin-layer chromatography;Cone;J Pharm Sci,1963

5. Structure of tubulin at 6.5 A and location of the taxol-binding site;Nogales;Nature,1995

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