Fragment-Based Design of Novel Quinazolinon Derivatives as Human Acrosin Inhibitors-Reference-Cited by-同舟云学术

Fragment-Based Design of Novel Quinazolinon Derivatives as Human Acrosin Inhibitors

Published:2013-03-28 Issue:4 Volume:81 Page:437-441
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Ning Weiwei¹,Zhu Ju¹,Zheng Canhui¹,Liu Xuefei¹,Song Yunlong¹,Zhou Youjun¹,Zhang Xiaomeng¹,Zhang Ling¹,Sheng Chunquan¹,Lv Jiaguo¹

Affiliation:

1. Department of medicinal Chemistry; School of Pharmacy; Second Military Medical University; 325 Guohe Road; Shanghai; 200433; China

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.12106/fullpdf

Reference18 articles.

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3. Proteinase inhibitors from the medicinal leech Hirudo medicinalis;Baskova;Biochemistry,2001

4. The effect of the trypsin inhibitor aprotinin (Trasylol) and TLCK on the gelatinolytic activity of acrosin and the motility of rabbit sperm in vitro;Pakzad;Z Mikrosk Anat Forsch,1989

5. Inhibition of sperm-zona binding by suramin, a potential ‘lead’ compound for design of new anti-fertility agents;Jones;Mol Hum Reprod,1996

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