Synthesis, Antidepressant Evaluation and Docking Studies of Long-Chain Alkylnitroquipazines as Serotonin Transporter Inhibitors-Reference-Cited by-同舟云学术

Synthesis, Antidepressant Evaluation and Docking Studies of Long-Chain Alkylnitroquipazines as Serotonin Transporter Inhibitors

Published:2013-04-11 Issue:6 Volume:81 Page:695-706
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Gabrielsen Mari¹,Wołosewicz Karol²,Zawadzka Anna³,Kossakowski Jerzy²,Nowak Gabriel,Wolak Małgorzata⁴,Stachowicz Katarzyna⁵,Siwek Agata⁴,Ravna Aina W.¹,Kufareva Irina⁶,Kozerski Lech,Bednarek Elżbieta⁷,Sitkowski Jerzy⁷,Bocian Wojciech⁷,Abagyan Ruben⁶,Bojarski Andrzej J.⁵,Sylte Ingebrigt¹,Chilmonczyk Zdzisław⁷

Affiliation:

1. Medical Pharmacology and Toxicology, Department of Medical Biology, Faculty of Health Sciences; University of Tromsø; 9037; Tromsø; Norway

2. Institute of Chemistry; University of Białystok; 1 Hurtowa Street; 15-399; Białystok; Poland

3. Department of Medicinal Chemistry; Warsaw Medical University; Oczki 3; 02-007; Warsaw; Poland

4. Department of Pharmacobiology; Jagiellonian University Medical College; Medyczna 9; 30-688; Kraków; Poland

5. Institute of Pharmacology; Polish Academy of Sciences; 12 Smętna Street; 31-343; Kraków; Poland

6. Skaggs School of Pharmacy and Pharmaceutical Sciences; 9500 Gilman Drive; MC 0747; La Jolla; CA; 92093-0747; USA

7. National Medicines Institute; 30/34 Chełmska Street; 00-725; Warsaw; Poland

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.12116/fullpdf

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4. Second-generation SSRIs: human monoamine transporter binding profile of escitalopram and R-fluoxetine;Owens;Biol Psychiatry,2001

5. Serotonin transporter inhibitors: synthesis and binding potency of 2′-methyl- and 3′-methyl-6-nitroquipazine;Gerdes;Bioorg Med Chem Lett,2000

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