A novel fluorescence‐based functional assay for human OATP1A2 and OATP1C1 identifies interaction between third‐generation P‐gp inhibitors and OATP1A2-Reference-Cited by-同舟云学术

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A novel fluorescence‐based functional assay for human OATP1A2 and OATP1C1 identifies interaction between third‐generation P‐gp inhibitors and OATP1A2

Published:2019-12-17 Issue:12 Volume:287 Page:2468-2485
ISSN:1742-464X
Container-title:The FEBS Journal
language:en
Short-container-title:FEBS J

Author:

Bakos Éva¹,Német Orsolya¹,Patik Izabel¹,Kucsma Nóra¹,Várady György²,Szakács Gergely¹³,Özvegy‐Laczka Csilla¹^ORCID

Affiliation:

1. Membrane Protein Research Group Institute of Enzymology Research Centre for Natural Sciences Hungarian Academy of Sciences Budapest Hungary

2. Laboratory of Molecular Cell Biology Institute of Enzymology Research Centre for Natural Sciences Hungarian Academy of Sciences Budapest Hungary

3. Institute of Cancer Research Medical University Vienna Wien Austria

Publisher

Wiley

Subject

Cell Biology,Molecular Biology,Biochemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1111/febs.15156

Reference62 articles.

1. Functional Expression of P-glycoprotein and Organic Anion Transporting Polypeptides at the Blood-Brain Barrier: Understanding Transport Mechanisms for Improved CNS Drug Delivery?

2. Delivery of Biologics Across the Blood–Brain Barrier with Molecular Trojan Horse Technology

3. The choroid plexus in health and in disease: dialogues into and out of the brain

4. Transport across the choroid plexus epithelium

5. Membrane transporter proteins: a challenge for CNS drug development;Girardin F;Dialogues Clin Neurosci,2006

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3. Dissimilar Effect of P-Glycoprotein and Breast Cancer Resistance Protein Inhibition on the Distribution of Erlotinib to the Retina and Brain in Humans and Mice;Molecular Pharmaceutics;2023-10-26

4. The fluorescence‐based competitive counterflow assay developed for organic anion transporting polypeptides 1A2, 1B1, 1B3 and 2B1 identifies pentamidine as a selective OATP1A2 substrate;The FASEB Journal;2023-10-02

5. Molecular Mechanisms of Organic Anion Transporting Polypeptide–Mediated Organic Anion Clearance at the Blood–Cerebrospinal Fluid Barrier;Molecular Pharmacology;2023-08-31

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