Inhibition of human CYP1 enzymes by a classical inhibitor α‐naphthoflavone and a novel inhibitor N ‐(3, 5‐dichlorophenyl)cyclopropanecarboxamide: An in vitro and in silico study-Reference-Cited by-同舟云学术

Inhibition of human CYP1 enzymes by a classical inhibitor α‐naphthoflavone and a novel inhibitor N ‐(3, 5‐dichlorophenyl)cyclopropanecarboxamide: An in vitro and in silico study

Published:2020-03-09 Issue:5 Volume:95 Page:520-533
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Juvonen Risto Olavi¹^ORCID,Jokinen Elmeri Matias²^ORCID,Javaid Adeel¹,Lehtonen Marko¹³,Raunio Hannu¹,Pentikäinen Olli Taneli²^ORCID

Affiliation:

1. Faculty of Health Sciences School of Pharmacy University of Eastern Finland Kuopio Finland

2. Faculty of Medicine, Integrative Physiology and Pharmacology Institute of Biomedicine University of Turku Turku Finland

3. LC‐MS Metabolomics Center Biocenter Kuopio Kuopio Finland

Funder

Academy of Finland

Sigrid Juséliuksen Säätiö

Varsinais-Suomen Rahasto

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1111/cbdd.13669

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5. Tight-binding inhibition by α-naphthoflavone of human cytochrome P450 1A2

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