Characterization of a Pyrazolo[4,3-d]pyrimidine Inhibitor of Cyclin-Dependent Kinases 2 and 5 and Aurora A With Pro-Apoptotic and Anti-Angiogenic ActivityIn Vitro

Author:

Řezníčková Eva1,Weitensteiner Sabine2,Havlíček Libor3,Jorda Radek1,Gucký Tomáš1,Berka Karel4,Bazgier Václav15,Zahler Stefan2,Kryštof Vladimír1,Strnad Miroslav1

Affiliation:

1. Laboratory of Growth Regulators & Department of Chemical Biology and Genetics; Centre of the Region Haná for Biotechnological and Agricultural Research; Palacký University and Institute of Experimental Botany AS CR; Šlechtitelů 27 78371 Olomouc Czech Republic

2. Department of Pharmacy; LMU Munich - Center for Drug Research - Pharmaceutical Biology; Butenandtstr. 5-13 81377 Munich Germany

3. Isotope Laboratory; Institute of Experimental Botany ASCR; Vídeňská 1083 14220 Prague Czech Republic

4. Regional Centre of Advanced Technologies and Materials; Department of Physical Chemistry; Faculty of Science; Palacký University; 17. listopadu 12 77146 Olomouc Czech Republic

5. Department of Physical Chemistry; Faculty of Science; Palacký University; 17. listopadu 1192/12 771 46 Olomouc Czech Republic

Funder

Grantová Agentura České Republiky

Ministry of Education, Youth and Sports of the Czech Republic

Internal Grant Agency of Palacký University

Deutsche Forschungsgemeinschaft

German Federal Ministry of Education and Research

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

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