Synthesis of Analogues of BCTC Incorporating a Pyrrolidinyl Linker and Biological Evaluation as Transient Receptor Potential Vanilloid 1 Antagonists-Reference-Cited by-同舟云学术

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Synthesis of Analogues of BCTC Incorporating a Pyrrolidinyl Linker and Biological Evaluation as Transient Receptor Potential Vanilloid 1 Antagonists

Published:2015-10-05 Issue:2 Volume:87 Page:306-311
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Yan Lin¹,Wang Jingjie²,Pan Miaobo²,Qiu Qianqian²,Huang Wenlong²,Qian Hai²

Affiliation:

1. Institute of Chemistry & Biology; Henan University; Kaifeng 475004 China

2. State Key Laboratory of Natural Medicines; Center of Drug Discovery; China Pharmaceutical University; 24 Tongjiaxiang Nanjing 210009 China

Funder

Natural Science Foundation of Jiangsu Province of China

Fundamental Research Funds for the Central Universities of China

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.12661/fullpdf

Reference30 articles.

1. The cloned capsaicin receptor integrates multiple pain-producing stimuli;Tominaga;Neuron,1998

2. Vanilloid receptors on sensory nerves mediate the vasodilator action of anandamide;Zygmunt;Nature,1999

3. An endogenous capsaicin-like substance with high potency at recombinant and native vanilloid VR1 receptors;Huang;Proc Natl Acad Sci USA,2002

4. AMG 9810 [(E)-3-(4-t-butylphenyl)-N-(2,3-dihydrobenzo[b][1,4] dioxin-6-yl)acrylamide], a novel vanilloid receptor 1 (TRPV1) antagonist with antihyperalgesic properties;Gavva;J Pharmacol Exp Ther,2005

5. Selective blockade of the capsaicin receptor TRPV1 attenuates bone cancer pain;Ghilardi;J Neurosci,2005

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