The structural conformation of the tachykinin domain drives the anti‐tumoural activity of an octopus peptide in melanoma BRAF V600E

Author:

Moral‐Sanz Javier1ORCID,Fernandez‐Rojo Manuel A.234ORCID,Colmenarejo Gonzalo5ORCID,Kurdyukov Sergey6,Brust Andreas7,Ragnarsson Lotten7ORCID,Andersson Åsa7,Vila Sabela F.18,Cabezas‐Sainz Pablo8,Wilhelm Patrick7ORCID,Vela‐Sebastián Ana1,Fernández‐Carrasco Isabel1,Chin Yanni K. Y.79,López‐Mancheño Yaiza2,Smallwood Taylor B.10,Clark Richard J.710ORCID,Fry Bryan G.11,King Glenn F.712ORCID,Ramm Grant A.313ORCID,Alewood Paul F.7ORCID,Lewis Richard J.7ORCID,Mulvenna Jason P.14,Boyle Glen M.15ORCID,Sanchez Laura E.8,Neely G. Gregory6ORCID,Miles John J.1617181920,Ikonomopoulou Maria P.1716ORCID

Affiliation:

1. Translational Venomics Group Madrid Institute for Advanced Studies in Food Madrid Spain

2. Hepatic Regenerative Medicine Group Madrid Institute for Advanced Studies in Food Madrid Spain

3. Hepatic Fibrosis Group, Department of Cell and Molecular Biology QIMR Berghofer Medical Research Institute Herston Queensland Australia

4. Diamantina Institute The University of Queensland St. Lucia Queensland Australia

5. Biostatistics & Bioinformatics Unit Madrid Institute for Advances Studies in Food Madrid Spain

6. Dr. John and Anne Chong Lab for Functional Genomics, Charles Perkins Centre, Centenary Institute, and School of Life and Environmental Sciences University of Sydney Camperdown New South Wales Australia

7. Institute for Molecular Bioscience The University of Queensland St Lucia Queensland Australia

8. Department of Zoology, Genetics and Physical Anthropology University of Santiago de Compostela Lugo Spain

9. Centre for Advanced Imaging The University of Queensland St Lucia Queensland Australia

10. School of Biomedical Sciences The University of Queensland St Lucia Queensland Australia

11. School of Biological Sciences The University of Queensland St Lucia Queensland Australia

12. Australian Research Council Centre of Excellence for Innovations in Peptide and Protein Science The University of Queensland Queensland Australia

13. Faculty of Medicine The University of Queensland Brisbane Queensland Australia

14. Infectious Diseases Program QIMR Berghofer Medical Research Institute Brisbane Queensland Australia

15. Department of Cell and Molecular Biology, Cancer Program QIMR Berghofer Medical Research Institute Brisbane Queensland Australia

16. Department of Immunology QIMR Berghofer Medical Research Institute Brisbane Queensland Australia

17. Centre for Biodiscovery and Molecular Development of Therapeutics and Centre for Biosecurity in Tropical Infectious Diseases James Cook University Cairns Queensland Australia

18. The Australian Institute of Tropical Health and Medicine (AITHM) James Cook University Cairns Queensland Australia

19. Centre for Molecular Therapeutics James Cook University Cairns Queensland Australia

20. Centre for Tropical Bioinformatics and Molecular Biology James Cook University Cairns Queensland Australia

Funder

Australian Research Council

Schweizerischer Nationalfonds zur Förderung der Wissenschaftlichen Forschung

Publisher

Wiley

Subject

Pharmacology

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