Pharmacological characterization of two novel and potent 5-HT4 receptor agonists, RS 67333 and RS 67506, in vitro and in vivo-Reference-Cited by-同舟云学术

Pharmacological characterization of two novel and potent 5-HT4 receptor agonists, RS 67333 and RS 67506, in vitro and in vivo

Published:1995-08 Issue:8 Volume:115 Page:1387-1392
ISSN:0007-1188
Container-title:British Journal of Pharmacology
language:en
Short-container-title:

Author:

Eglen R.M.,Bonhaus D.W.,Johnson L.G.,Leung E.,Clark R.D.

Publisher

Wiley

Subject

Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1476-5381.1995.tb16628.x/fullpdf

Reference27 articles.

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2. 5-Hydroxytryptamine4 receptors mediate relaxation of the rat oesophageal tunica muscularis mucosae;BAXTER;Naunyn-Schmied. Arch. Pharmacol.,1991

3. 5-HT4 receptors: potential therapeutic implications in neurology and psychiatry;BOCKAERT;CNS Drugs,1994

4. [3H] RS 23597-190, a potent 5-hydroxytryptamine4 antagonist labels sigma-1 but not sigma2 binding sites in guinea-pig brain;BONHAUS;J. Pharmacol. Exp. Ther.,1994

5. Relationship between inhibitor constant (Ki) and the concentration of inhibitor which causes 50 percent inhibition (IC50) of an enzymatic reaction;CHENG;Biochem. Pharmacol.,1973

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