Desensitization and functional antagonism by β-adrenoceptor and muscarinic receptor agonists, respectively: a comparison with receptor alkylation for calculation of apparent agonist affinity-Reference-Cited by-同舟云学术

Desensitization and functional antagonism by β-adrenoceptor and muscarinic receptor agonists, respectively: a comparison with receptor alkylation for calculation of apparent agonist affinity

Published:1991-08 Issue:4 Volume:103 Page:1951-1957
ISSN:0007-1188
Container-title:British Journal of Pharmacology
language:en
Short-container-title:

Author:

Eglen R.M.,Montgomery W.W.,Whiting R.L.

Publisher

Wiley

Subject

Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1476-5381.1991.tb12358.x/fullpdf

Reference40 articles.

1. Variable receptor affinity hypothesis;BEVAN;FASEB J.,1989

2. Pharmacological analysis of β-adrenoceptor-mediated agonism in the guinea-pig isolated, right atrium;BLACK;Br. J. Pharmacol.,1985

3. Functional antagonism as a means of determining dissociation constants and relative efficacies of sympathomimetic amines in guinea-pig isolated atria;BROADLEY;Br. J. Pharmacol.,1979

4. On the use of functional antagonism to estimate dissociation constants for beta adrenergic receptor agonists in isolated guinea-pig trachea;BUCKNER;J. Pharmacol. Exp. Ther.,1975

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1. Relationship between desensitization and downregulation of beta-adrenoceptors in cardiac tissues after prolonged in vivo infusion of T-0509, a beta(1)-adrenoceptor agonist;JPN J PHARMACOL;1997

2. Relationship between Desensitization and Downregulation of β-Adrenoceptors in Cardiac Tissues after Prolonged In Vivo Infusion of T-0509, a β1-Adrenoceptor Agonist;Japanese Journal of Pharmacology;1997

3. Interactions between responses mediated by activation of adenosine A2 receptors and α1-adrenoceptors in the rabbit isolated aorta;British Journal of Pharmacology;1993-06

4. Alprenolol and Bromoacetylalprenololmenthane are Competitive Slowly Reversible Antagonists at the β1-Adrenoceptors of Rat Left Atria;Journal of Cardiovascular Pharmacology;1993-01