Novel opioid cyclic tetrapeptides: Trp isomers of CJ-15,208 exhibit distinct opioid receptor agonism and short-acting κ opioid receptor antagonism

Author:

Ross Nicolette C,Reilley Kate J,Murray Thomas F,Aldrich Jane V,McLaughlin Jay P

Publisher

Wiley

Subject

Pharmacology

Reference53 articles.

1. Peptide kappa opioid receptor ligands: potential for drug development;Aldrich;AAPS J,2009

2. Aldrich JV Patkar KA Chappa AK Fang W Audus KL Lunte SM et al 2007 Development of centrally acting peptide analogs: structural transport studies and pharmacological evaluation of analogs of the opioid peptide dynorphin A Proceedings of the 4th International Peptide Symposium http://www.peptideoz.org/docs/M_64_Jane_Aldrich.pdf

3. Zyklophin, a systemically active selective kappa opioid receptor peptide antagonist with short duration of action;Aldrich;Proc Natl Acad Sci USA,2009

4. Synthesis and opioid activity of conformationally constrained dynorphin A analogues. 2. Conformational constraint in the ‘address’ sequence;Arttamangkul;J Med Chem,1997

5. Some quantitative uses of drug antagonists;Arunlakshana;Br J Pharmacol Chemother,1959

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