Slow receptor dissociation is not a key factor in the duration of action of inhaled long-acting β2-adrenoceptor agonists
Author:
Publisher
Wiley
Subject
Pharmacology
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1476-5381.2011.01639.x/fullpdf
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4. A physical properties based approach for the exploration of a 4-hydroxybenzothiazolone series of beta2-adrenoceptor agonists as inhaled long-acting bronchodilators;Beattie;Bioorg Med Chem Lett,2010
5. The short, the long and the ‘ultra-long’: why duration of bronchodilator action matters in chronic obstructive pulmonary disease;Beeh;Adv Ther,2010
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