The physiological relevance of low agonist affinity binding at opioid μ-receptors-Reference-Cited by-同舟云学术

The physiological relevance of low agonist affinity binding at opioid μ-receptors

Published:1988-06 Issue:2 Volume:94 Page:625-631
ISSN:0007-1188
Container-title:British Journal of Pharmacology
language:en
Short-container-title:

Author:

Carroll Jacqueline A.,Shaw John S.,Wickenden Alan D.

Publisher

Wiley

Subject

Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1476-5381.1988.tb11569.x/fullpdf

Reference22 articles.

1. Interaction of ligands with the opiate receptor of brain membranes: Regulation by ions and nucleotides;BLUME;Proc. Natl. Acad. Sci. U.S.A.,1978

2. Mu receptor binding in physiological media: Comparison with isolated tissue data;CARROLL;Neuropeptides,1984

3. Multiple opiate receptors: Different regional distribution in the brain and differential binding of opiate and opioid peptides;CHANG;Mol. Pharmacol,1979

4. Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50% inhibition (150) of an enzymatic reaction;CHENG;Biochem. Pharmacol,1973

5. Receptor binding and pharmacological activity of opiates in the guinea-pig intestine;CREESE;J. Pharmacol. Exp. Ther,1975

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