Pharmacologically distinct phenotypes of α1B-adrenoceptors: variation in binding and functional affinities for antagonists

Author:

Yoshiki Hatsumi1,Uwada Junsuke12,Anisuzzaman Abu Syed Md1,Umada Hidenori1,Hayashi Ryoji3,Kainoh Mie3,Masuoka Takayoshi4,Nishio Matomo4,Muramatsu Ikunobu1245

Affiliation:

1. Division of Pharmacology, Department of Biochemistry and Bioinformative Sciences, School of Medicine; University of Fukui; Eiheiji Fukui Japan

2. Organization for Life Science Advancement Programs; University of Fukui; Eiheiji Fukui Japan

3. Pharmaceutical Research Laboratories; Toray Industries, Inc.; Kamakura Kanagawa Japan

4. Department of Pharmacology, School of Medicine; Kanazawa Medical University; Uchinada Ishikawa Japan

5. Kimura Hospital; Awara Fukui Japan

Funder

Ministry of Education, Culture, Sports, Science and Technology of Japan

Smoking Research Foundation of Japan

Organization for Life Science Advancement Programs (Research and Education Program for Life Science, Translational Research Program

Life Science Research Laboratory, University of Fukui

Publisher

Wiley

Subject

Pharmacology

Reference43 articles.

1. The Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptors;Alexander;Br J Pharmacol.,2013

2. Influence of tissue integrity on pharmacological phenotypes of muscarinic acetylcholine receptors in the rat cerebral cortex;Anisuzzaman;J Pharmacol Exp Ther,2011

3. Novel contribution of cell surface and intracellular M1-muscarinic acetylcholine receptors to synaptic plasticity in hippocampus;Anisuzzaman;J Neurochem,2013

4. β3-Adrenoceptor agonists: potential. pitfalls and progress;Arch;Eur J Pharmacol,2002

5. Some quantitative uses of drug antagonists;Arunlakshana;Br J Pharmacol Chemother,1959

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