Towards Development of a Dermal Pain Model:In VitroActivation of Rat and Human Transient Receptor Potential Ankyrin Repeat 1 and Safe Dermal Injection ofo-Chlorobenzylidene Malononitrile to Rat

Author:

Annas Anita1,Berg Anna-Lena12,Nyman Eva34,Meijer Thomas56,Lundgren Viveka5,Franzén Bo37,Ståhle Lars89

Affiliation:

1. Global Safety Assessment; AstraZeneca R&D; Södertälje Sweden

2. Medical Products Agency; Uppsala Sweden

3. Neuroscience, Innovative Medicines CNS/Pain; AstraZeneca R&D; Södertälje Sweden

4. The National Board of Health and Welfare; Stockholm Sweden

5. Pharmaceutical Development, Medicines Evaluation CNS/Pain; AstraZeneca R&D; Södertälje Sweden

6. SP Process Development; Södertälje Sweden

7. Cancer Center Karolinska; Karolinska Institute and Hospital; Stockholm Sweden

8. Clinical Sciences, Neuroscience Therapeutic Area; AstraZeneca R&D; Södertälje Sweden

9. Pain Clinic; Karolinska Hospital Huddinge and CLINTEC Karolinska Institute; Stockholm Sweden

Funder

AstraZeneca

Publisher

Wiley

Subject

Pharmacology,Toxicology,General Medicine

Reference28 articles.

1. Jonzon B Sundgren-Andersson A Quiding H Carlsson M Segerdahl M Karin A Target validation and dose response study using intradermal microgram doses of TRPV1 antagonists in healthy volunteers IASP Montreal, QC 2010

2. TRP channels;Venkatachalam;Annu Rev Biochem,2007

3. 4-Hydroxynonenal, an endogenous aldehyde, causes pain and neurogenic inflammation through activation of the irritant receptor TRPA1;Trevisani;Proc Natl Acad Sci USA,2007

4. TRPA1: A transducer and amplifier of pain and inflammation;Koivisto;Basic Clin Pharmacol Toxicol,2014

5. Mustard oils and cannabinoids excite sensory nerve fibres through the TRP channel ANKTM1;Jordt;Nature,2004

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