Aporphinoid Antagonists of 5-HT2AReceptors: Further Evaluation of Ring A Substituents and the Size of Ring C-Reference-Cited by-同舟云学术

登录注册会员服务联系我们

Aporphinoid Antagonists of 5-HT2AReceptors: Further Evaluation of Ring A Substituents and the Size of Ring C

Published:2014-06-03 Issue:5 Volume:84 Page:558-566
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Ponnala Shashikanth¹,Kapadia Nirav¹²,Navarro Hernán A.³,Harding Wayne W.¹²

Affiliation:

1. Chemistry Department; Hunter College; CUNY; 695 Park Avenue NY 10065 USA

2. The Graduate Center; City University of New York; 365 5th Ave. NY 10016 USA

3. Center for Organic and Medicinal Chemistry; Research Triangle Institute; Research Triangle Park; NC 27709 USA

Funder

National Institutes of Health

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.12345/fullpdf

Reference33 articles.

1. Cytotoxic and antimicrobial activities of aporphine alkaloids isolated from Stephania venosa (Blume) Spreng;Makarasen;Planta Med,2011

2. Cytotoxicity of aporphines in human colon cancer cell lines HCT-116 and Caco-2: an SAR study;Ponnala;Bioorg Med Chem Lett,2011

3. Cytotoxic aporphine alkaloids from Ocotea acutifolia;Garcez;Planta Med,2011

4. Antiplasmodial activity of aporphine alkaloids and sesquiterpene lactones from Liriodendron tulipifera L;Graziose;J Ethnopharmacol,2011

5. Cytotoxic and antitumor potentialities of aporphinoid alkaloids;Stevigny;Curr Med Chem Anticancer Agents,2005

Cited by 7 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Structure-activity relationship study of 4,5-didehydroguadiscine, an aporphine alkaloid showing potent melanogenesis-inhibitory activity in B16 melanoma cells;Bioorganic & Medicinal Chemistry Letters;2022-12

2. Semisynthetic Transformations on (+)-Boldine Reveal a 5-HT_2A/2CR Antagonist;Journal of Natural Products;2022-08-24

3. Mechanism Exploration of Arylpiperazine Derivatives Targeting the 5-HT2A Receptor by In Silico Methods;Molecules;2017-06-26

4. Synthesis and evaluation of aporphine analogs containing C1 allyl isosteres at the h5-HT2A receptor;Bioorganic & Medicinal Chemistry Letters;2015-11

5. C4 phenyl aporphines with selective h5-HT2B receptor affinity;Bioorganic & Medicinal Chemistry Letters;2015-09

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号京ICP备18003416号-3