Further Insights Into the Pharmacology of the Human Trace Amine-Associated Receptors: Discovery of Novel Ligands for TAAR1 by a Virtual Screening Approach-Reference-Cited by-同舟云学术

Further Insights Into the Pharmacology of the Human Trace Amine-Associated Receptors: Discovery of Novel Ligands for TAAR1 by a Virtual Screening Approach

Published:2014-06-30 Issue:6 Volume:84 Page:712-720
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Cichero Elena¹,Espinoza Stefano²,Franchini Silvia³,Guariento Sara¹,Brasili Livio³,Gainetdinov Raul R.²⁴⁵,Fossa Paola¹

Affiliation:

1. Dipartimento di Farmacia; Università degli Studi di Genova; Viale Benedetto XV n. 3 Genova 16132 Italy

2. Department of Neuroscience and Brain Technologies; Istituto Italiano di Tecnologia; Via Morego 30, Genova 16163 Italy

3. Dipartimento di Scienze della Vita; Università degli Studi di Modena e Reggio Emilia; Via Campi 183 Modena 41100 Italy

4. Skolkovo Institute of Science and Technology; Skolkovo Moscow Region 143025 Russia

5. Faculty of Biology and Soil Science; St. Petersburg State University; St. Petersburg 199034 Russia

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.12367/fullpdf

Reference26 articles.

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2. Trace amine-associated receptors as emerging therapeutic targets;Sotnikova;Mol Pharmacol,2009

3. Trace amines: identification of a family of mammalian G protein-coupled receptors;Borowsky;Proc Natl Acad Sci USA,2001

4. Trace amine-associated receptor 1 as a monoaminergic modulator in brain;Xie;Biochem Pharmacol,2009

5. Normal thermoregulatory responses to 3-iodothyronamine, trace amines and amphetamine-like psychostimulants in trace amine associated receptor 1 knockout mice;Panas;J Neurosci Res,2010

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