Pharmacological characterization ofN-[(2S)-5-(6-fluoro-3-pyridinyl)-2, 3-dihydro-1H-inden-2-yl]-2-propanesulfonamide: a novel, clinical AMPA receptor positive allosteric modulator-Reference-Cited by-同舟云学术

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Pharmacological characterization ofN-[(2S)-5-(6-fluoro-3-pyridinyl)-2, 3-dihydro-1H-inden-2-yl]-2-propanesulfonamide: a novel, clinical AMPA receptor positive allosteric modulator

Published:2017-01-31 Issue:5 Volume:174 Page:370-385
ISSN:0007-1188
Container-title:British Journal of Pharmacology
language:en
Short-container-title:British Journal of Pharmacology

Author:

Ward Simon E¹²,Beswick Paul¹,Calcinaghi Novella³,Dawson Lee A²,Gartlon Jane²,Graziani Francesca³,Jones Declan N C²,Lacroix Laurent²⁴,Selina Mok M H²,Oliosi Beatrice³,Pardoe Joanne²,Starr Kathryn²,Woolley Marie L²,Harries Mark H²

Affiliation:

1. University of Sussex; Brighton UK

2. Neurosciences Centre of Excellence for Drug Discovery; GlaxoSmithKline; Harlow UK

3. Neurosciences Centre of Excellence for Drug Discovery; GlaxoSmithKline Medicines Research Centre; Verona Italy

4. Health Sciences Research Center, Whiteland's College; University of Roehampton; London UK

Publisher

Wiley

Subject

Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/bph.13696/fullpdf

Reference52 articles.

1. Editing for an AMPA receptor subunit RNA in prefrontal cortex and striatum in Alzheimer's disease, Huntington's disease and schizophrenia;Akbarian;Brain Res,1995

2. The Concise Guide to PHARMACOLOGY 2015/16: Ligand-gated ion channels;Alexander;Br J Pharmacol,2015

3. Effects of a centrally active benzoylpyrrolidine drug on AMPA receptor kinetics;Arai;Neuroscience,1996

4. Dynamics of the ligand binding domain layer during AMPA receptor activation;Baranovic;Biophys J,2016

5. Expression of transcripts encoding AMPA receptor subunits and associated postsynaptic proteins in the macaque brain;Beneyto;J Comp Neurol,2004

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