Pharmacological and SAR analysis of the LINS01 compounds at the human histamine H1 , H2 , and H3 receptors-Reference-Cited by-同舟云学术

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Pharmacological and SAR analysis of the LINS01 compounds at the human histamine H1 , H2 , and H3 receptors

Published:2018-09-24 Issue:1 Volume:93 Page:89-95
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Corrêa Michelle Fidelis¹,Barbosa Álefe Jhonatas Ramos¹,Fernandes Gustavo Ariel Borges¹,Baker Jillian G.²,Fernandes João Paulo dos Santos¹^ORCID

Affiliation:

1. Departamento de Ciências Farmacêuticas; Universidade Federal de São Paulo; Diadema Brazil

2. Cell Signalling Research Group; School of Life Sciences; University of Nottingham; Nottingham UK

Funder

Conselho Nacional de Desenvolvimento Científico e Tecnológico

Fundação de Amparo à Pesquisa do Estado de São Paulo

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.13387/fullpdf

Reference27 articles.

1. International Union of Basic and Clinical Pharmacology. XCVIII. Histamine Receptors

2. Histamine H4 Receptor Ligands: Future Applications and State of Art

3. Heteroreceptor Complexes Formed by Dopamine D1, Histamine H3, and N-Methyl-D-Aspartate Glutamate Receptors as Targets to Prevent Neuronal Death in Alzheimer’s Disease

4. Neuronal histamine and cognitive symptoms in Alzheimer's disease

5. The Histamine H3 Receptor: Structure, Pharmacology, and Function

Cited by 7 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Therapeutic potential of LINS01 histamine H3 receptor antagonists as antineoplastic agents for triple negative breast cancer;Biomedicine & Pharmacotherapy;2024-05

2. The histamine H4 receptor antagonist 1-[(5-chloro-2,3-dihydro-1-benzofuran-2-yl)methyl]-4-methyl-piperazine(LINS01007) prevents the development of DSS-induced colitis in mice;International Immunopharmacology;2024-05

3. Evaluation of the histamine H ₃ receptor antagonists from LINS01 series as cholinesterases inhibitors: Enzymatic and modeling studies;Chemical Biology & Drug Design;2022-09-08

4. Novel potent (dihydro)benzofuranyl piperazines as human histamine receptor ligands – Functional characterization and modeling studies on H3 and H4 receptors;Bioorganic & Medicinal Chemistry;2021-01

5. Novel potent vasodilating agents: Evaluation of the activity and potency of LINS01005 and derivatives in rat aorta;European Journal of Pharmaceutical Sciences;2020-02

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