Synthesis of acyl derivatives of thiazolo[5.4-b]indole-Reference-Cited by-同舟云学术

Synthesis of acyl derivatives of thiazolo[5.4-b]indole

Published:2019-12-06 Issue:4 Volume:55 Page:436-441
ISSN:2524-2342
Container-title:Proceedings of the National Academy of Sciences of Belarus, Chemical Series
language:
Short-container-title:Vescì Akademìì navuk Belarusì. Seryâ himičnyh navuk

Author:

Lopatik D. V.¹,Kuvaeva Z. I.¹,Bondareva O. M.¹,Naidenov V. E.¹,Tychinskaya L. Yu.¹

Affiliation:

1. Institute of Physical Organic Chemistry of the National Academy of Sciences of Belarus

Abstract

2-Amino-4-acetylthiazolo[5,4-b]indole and its bromosubstituted analogue contain a free amino group and are initial compounds for chemical modification in order to obtain on their basis functional derivatives having high therapeutic activity. By the interaction of these 2-aminо-4-acetylthiazolo[5,4-b]indoles with succinic and maleic anhydrides, the corresponding imides and amides were obtained, which are of interest for use in order to create on their basis antihypoxic and actoprotective agents.

Publisher

Publishing House Belorusskaya Nauka

Subject

Inorganic Chemistry,Organic Chemistry,Chemistry (miscellaneous),Analytical Chemistry

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