Discovery of PDK1 Kinase Inhibitors with a Novel Mechanism of Action by Ultrahigh Throughput Screening-Reference-Cited by-同舟云学术

Discovery of PDK1 Kinase Inhibitors with a Novel Mechanism of Action by Ultrahigh Throughput Screening

Published:2010-06 Issue:24 Volume:285 Page:18838-18846
ISSN:0021-9258
Container-title:Journal of Biological Chemistry
language:en
Short-container-title:Journal of Biological Chemistry

Author:

Bobkova Ekaterina V.,Weber Michael J.,Xu Zangwei,Zhang Yan-Ling,Jung Joon,Blume-Jensen Peter,Northrup Alan,Kunapuli Priya,Andersen Jannik N.,Kariv Ilona

Publisher

Elsevier BV

Subject

Cell Biology,Molecular Biology,Biochemistry

Reference38 articles.

1. The Protein Kinase Complement of the Human Genome

2. The Current Status of Drug Discovery Against the Human Kinome

3. Global, In Vivo, and Site-Specific Phosphorylation Dynamics in Signaling Networks

4. A quantitative atlas of mitotic phosphorylation

5. Wild-Type BRAF Is Required for Response to Panitumumab or Cetuximab in Metastatic Colorectal Cancer

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