The Kinetic Factors That Determine the Affinity and Selectivity for Slow Binding Inhibition of Human Prostaglandin H Synthase 1 and 2 by Indomethacin and Flurbiprofen-Reference-Cited by-同舟云学术

The Kinetic Factors That Determine the Affinity and Selectivity for Slow Binding Inhibition of Human Prostaglandin H Synthase 1 and 2 by Indomethacin and Flurbiprofen

Published:1996-02 Issue:7 Volume:271 Page:3548-3554
ISSN:0021-9258
Container-title:Journal of Biological Chemistry
language:en
Short-container-title:Journal of Biological Chemistry

Author:

Callan Ondine Harris,So On-Yee,Swinney David C.

Publisher

Elsevier BV

Subject

Cell Biology,Molecular Biology,Biochemistry

Reference22 articles.

1. Inhibition of Prostaglandin Synthesis as a Mechanism of Action for Aspirin-like Drugs

2. Expression of a mitogen-responsive gene encoding prostaglandin synthase is regulated by mRNA splicing.

3. Inducible isoforms of cyclooxygenase and nitric-oxide synthase in inflammation.

4. Mitogen-inducible prostaglandin G/H synthase: A new target for nonsteroidal antiinflammatory drugs

5. Selectivity of nonsteroidal antiinflammatory drugs as inhibitors of constitutive and inducible cyclooxygenase.

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