Physiologically relevant orthogonal assays for the discovery of small-molecule modulators of WIP1 phosphatase in high-throughput screens-Reference-Cited by-同舟云学术

登录注册会员服务联系我们

Physiologically relevant orthogonal assays for the discovery of small-molecule modulators of WIP1 phosphatase in high-throughput screens

Published:2019-11 Issue:46 Volume:294 Page:17654-17668
ISSN:0021-9258
Container-title:Journal of Biological Chemistry
language:en
Short-container-title:Journal of Biological Chemistry

Author:

Clausse Victor,Tao Dingyin^ORCID,Debnath Subrata,Fang Yuhong^ORCID,Tagad Harichandra D.^ORCID,Wang Yuhong,Sun Hongmao,LeClair Christopher A.^ORCID,Mazur Sharlyn J.^ORCID,Lane Kelly,Shi Zhen-Dan,Vasalatiy Olga,Eells Rebecca,Baker Lynn K.,Henderson Mark J.^ORCID,Webb Martin R.,Shen Min^ORCID,Hall Matthew D.^ORCID,Appella Ettore,Appella Daniel H.,Coussens Nathan P.^ORCID

Funder

HHS | NIH | National Cancer Institute

HHS | NIH | National Center for Advancing Translational Sciences

Cancer Research UK

UK Research and Innovation | Medical Research Council

Wellcome Trust

HHS | NIH | National Heart, Lung, and Blood Institute

HHS | NIH | National Institute of Diabetes and Digestive and Kidney Diseases

Publisher

Elsevier BV

Subject

Cell Biology,Molecular Biology,Biochemistry

Reference79 articles.

1. Genomics and evolution of protein phosphatases;Chen;Sci. Signal,2017

2. Therapeutic targeting of oncogenic tyrosine phosphatases;Frankson;Cancer Res,2017

3. Tumor suppressive protein phosphatases in human cancer: emerging targets for therapeutic intervention and tumor stratification;Meeusen;Int. J. Biochem. Cell Biol,2018

4. Challenges and opportunities in the development of protein phosphatase-directed therapeutics;De Munter;ACS Chem. Biol,2013

5. New approaches to difficult drug targets: the phosphatase story;Lazo;SLAS Discov,2017

Cited by 7 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Crystal structure and mechanistic studies of the PPM1D serine/threonine phosphatase catalytic domain;Journal of Biological Chemistry;2024-08

2. High-Throughput Capillary Liquid Chromatography Using a Droplet Injection and Application to Reaction Screening;Analytical Chemistry;2024-03-05

3. Use of in vitro methods combined with in silico analysis to identify potential skin sensitizers in the Tox21 10K compound library;Frontiers in Toxicology;2024-02-28

4. Alkyl-substituted N-methylaryl-N′-aryl-4-aminobenzamides: A new series of small molecule inhibitors for Wip1 phosphatase;European Journal of Medicinal Chemistry;2022-12

5. Discovery of Novel Small-Molecule Scaffolds for the Inhibition and Activation of WIP1 Phosphatase from a RapidFire Mass Spectrometry High-Throughput Screen;ACS Pharmacology & Translational Science;2022-09-28

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号京ICP备18003416号-3