Phosphomimetic substitution at Ser-33 of the chloroquine resistance transporter PfCRT reconstitutes drug responses in Plasmodium falciparum
Author:
Funder
Agence Nationale de la Recherche (ANR)
Deutsche Forschungsgemeinschaft (DFG)
PHC PROCOPE
Publisher
Elsevier BV
Subject
Cell Biology,Molecular Biology,Biochemistry
Reference55 articles.
1. Association of a novel mutation in the Plasmodium falciparum chloroquine resistance transporter with decreased piperaquine sensitivity;Agrawal;J. Infect. Dis,2017
2. A variant pfcrt isoform can contribute to Plasmodium falciparum resistance to the first-line partner drug piperaquine;Dhingra;MBio,2017
3. A critical role for PfCRT K76T in Plasmodium falciparum verapamil-reversible chloroquine resistance;Lakshmanan;EMBO J,2005
4. Evidence for a central role for pfcrt in conferring Plasmodium falciparum resistance to diverse antimalarial agents;Johnson;Mol. Cell,2004
5. Geographic patterns of Plasmodium falciparum drug resistance distinguished by differential responses to amodiaquine and chloroquine;Sá;Proc. Natl. Acad. Sci. U.S.A,2009
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1. Post-Translational Modifications of Proteins of Malaria Parasites during the Life Cycle;International Journal of Molecular Sciences;2024-06-02
2. Epitope specific antibodies to N- and C cytoplasmic domains of the Plasmodium falciparum chloroquine resistance transporter (PfCRT) differentiate native and post-translationally modified variant;Biochemical and Biophysical Research Communications;2023-08
3. PfCRT mutations conferring piperaquine resistance in falciparum malaria shape the kinetics of quinoline drug binding and transport;PLOS Pathogens;2023-06-07
4. A Plasmodium falciparum RING Finger E3 Ubiquitin Ligase Modifies the Roles of PfMDR1 and PfCRT in Parasite Drug Responses;Antimicrobial Agents and Chemotherapy;2023-02-16
5. The Knock-Down of the Chloroquine Resistance Transporter PfCRT Is Linked to Oligopeptide Handling in Plasmodium falciparum;Microbiology Spectrum;2022-08-31
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