Slow isomerization step in the interaction between mouse dopamine transporter and dopamine re-uptake inhibitor N-(3-iodoprop-2E-enyl)-2β-carbo-[3H]methoxy-3β-(4′-methylphenyl)nortropane
Author:
Publisher
Elsevier BV
Subject
General Neuroscience
Reference16 articles.
1. Synthesis, ligand binding, QSAR, and CoMFA study of 3β-(p-substituted phenyl)tropane-2β-carboxylic acid methyl esters;Carroll;J. Med. Chem.,1991
2. Synthesis and Ligand Binding of Nortropane Derivatives: N-Substituted 2β-Carbomethoxy-3β-(4‘-iodophenyl)nortropane and N-(3-Iodoprop-(2E)-enyl)-2β-carbomethoxy-3β-(3‘,4‘-disubstituted phenyl)nortropane. New High-Affinity and Selective Compounds for the Dopamine Transporter
3. PET study of [11C]β-CIT binding to monoamine transporters in the monkey and human brain;Farde;Synapse,1994
4. Pharmacogenetics of monoamine transporters;Glatt;Pharmacogenomics,2003
5. Synthesis and characteristic of radioiodonated N-(3-iodopropen-1-yl)-2β-carbomethoxy-3β-(4-chlorophenyl)tropanes: potential dopamine reuptake site imaging agents;Goodman;J. Med. Chem.,1994
Cited by 11 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Dopamine transporter interaction with blockers and transportable substrates: insights from kinetics study;Proceedings of the Estonian Academy of Sciences;2023
2. Inhibition of ligand–protein complex isomerization by some dopamine transporter inhibitors;Proceedings of the Estonian Academy of Sciences;2023
3. In Vitro Ligand Binding Kinetics Explains the Pharmacokinetics of [18F]FE-PE2I in Dopamine Transporter PET Imaging;ACS Medicinal Chemistry Letters;2018-11-29
4. Small Structural Changes at theN‐position of the Tropane Core Control the Mechanism of Nortropane Derivatives Binding to Dopamine Transporter;ChemistrySelect;2018-06-20
5. Kinetic tools for the identification of ligand–receptor interaction mechanisms;Proceedings of the Estonian Academy of Sciences;2017
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3