Low nanomolar GABA effects at extrasynaptic α4β1/β3δ GABAA receptor subtypes indicate a different binding mode for GABA at these receptors-Reference-Cited by-同舟云学术

Low nanomolar GABA effects at extrasynaptic α4β1/β3δ GABAA receptor subtypes indicate a different binding mode for GABA at these receptors

Published:2012-08 Issue:4 Volume:84 Page:549-557
ISSN:0006-2952
Container-title:Biochemical Pharmacology
language:en
Short-container-title:Biochemical Pharmacology

Author:

Karim Nasiara,Wellendorph Petrine,Absalom Nathan,Bang Line Haunstrup,Jensen Marianne Lerbech,Hansen Maja Michelle,Lee Ho Joon,Johnston Graham A.R.,Hanrahan Jane R.,Chebib Mary

Publisher

Elsevier BV

Subject

Pharmacology,Biochemistry

Reference48 articles.

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3. GABAA receptor ɛ and θ subunits display unusual structural variation between species and are enriched in the rat locus ceruleus;Sinkkonen;J Neurosci,2000

4. Extrasynaptic GABAA receptors: form, pharmacology, and function;Belelli;J Neurosci,2009

5. Pharmacological characterization of agonists at delta-containing GABAA receptors: functional selectivity for extrasynaptic receptors is dependent on the absence of gamma2;Storustovu;J Pharmacol Exp Ther,2006

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