Structure-based design and in vivo anti-arthritic activity evaluation of a potent dipeptidyl cyclopropyl nitrile inhibitor of cathepsin C-Reference-Cited by-同舟云学术

Structure-based design and in vivo anti-arthritic activity evaluation of a potent dipeptidyl cyclopropyl nitrile inhibitor of cathepsin C

Published:2019-06 Issue: Volume:164 Page:349-367
ISSN:0006-2952
Container-title:Biochemical Pharmacology
language:en
Short-container-title:Biochemical Pharmacology

Author:

Korkmaz Brice,Lesner Adam,Wysocka Magdalena,Gieldon Artur,Håkansson Maria,Gauthier Francis,Logan Derek T.,Jenne Dieter E.,Lauritzen Conni,Pedersen John

Funder

Unizyme

Ministère de l'Enseignement Supérieur et de la Recherche

Région Centre

National Science Center Poland

Publisher

Elsevier BV

Subject

Pharmacology,Biochemistry

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4. Dipeptidyl peptidase I: importance of progranzyme activation sequences, other dipeptide sequences, and the N-terminal amino group of synthetic substrates for enzyme activity;Tran;Arch. Biochem. Biophys.,2002

5. Dipeptidyl peptidase I activates neutrophil-derived serine proteases and regulates the development of acute experimental arthritis;Adkison;J. Clin. Invest.,2002

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