Glycine substitution of α1F64 residue at the loop D of GABAA receptor impairs gating – Implications for importance of binding site-channel gate linker rigidity-Reference-Cited by-同舟云学术

Glycine substitution of α1F64 residue at the loop D of GABAA receptor impairs gating – Implications for importance of binding site-channel gate linker rigidity

Published:2021-10 Issue: Volume:192 Page:114668
ISSN:0006-2952
Container-title:Biochemical Pharmacology
language:en
Short-container-title:Biochemical Pharmacology

Author:

Kłopotowski Karol^ORCID,Czyżewska Marta M.,Mozrzymas Jerzy W.^ORCID

Publisher

Elsevier BV

Subject

Pharmacology,Biochemistry

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2. Mutation of valine 53 at the interface between extracellular and transmembrane domains of the β2 principal subunit affects the GABAA receptor gating;European Journal of Pharmacology;2023-05

3. GABAA receptor proline 273 at the interdomain interface of the β2 subunit regulates entry into desensitization and opening/closing transitions;Life Sciences;2022-11

4. α₁ Proline 277 Residues Regulate GABA_AR Gating through M2-M3 Loop Interaction in the Interface Region;ACS Chemical Neuroscience;2022-10-11