Thermodynamics and kinetics of inhibitor binding to human equilibrative nucleoside transporter subtype-1
Author:
Funder
Biocenter Oulu/University of Oulu
Academy of Finland
Sigrid Juselius Foundation
FP7 Marie Curie European Reintegration Grant
Publisher
Elsevier BV
Subject
Pharmacology,Biochemistry
Reference38 articles.
1. Functional production and reconstitution of the human equilibrative nucleoside transporter (hENT1) in Saccharomyces cerevisiae. Interaction of inhibitors of nucleoside transport with recombinant hENT1 and a glycosylation-defective derivative (hENT1/N48Q);Vickers;Biochem. J.,1999
2. Equilibrative-sensitive nucleoside transporter and its role in gemcitabine sensitivity;Rauchwerger;Cancer Res.,2000
3. Allosteric binding of nucleoside triphosphates to RNA polymerase regulates transcription elongation;Foster;Cell,2001
4. Advances in the development of nucleoside and nucleotide analogues for cancer and viral diseases;Jordheim;Nat. Rev. Drug Discov.,2013
5. The equilibrative nucleoside transporter family, SLC29;Baldwin;Pflugers Arch.,2004
Cited by 12 articles. 订阅此论文施引文献 订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献
1. Exploring novel dilazep derivatives as hENT1 inhibitors and potentially covalent molecular tools;Purinergic Signalling;2024-06-15
2. A miniaturized mode-of-action profiling platform enables high throughput characterization of the molecular and cellular dynamics of EZH2 inhibition;Scientific Reports;2024-01-19
3. Kinetic profiling of novel spirobenzo-oxazinepiperidinone derivatives as equilibrative nucleoside transporter 1 inhibitors;Purinergic Signalling;2023-07-10
4. Novel variants provide differential stabilisation of human equilibrative nucleoside transporter 1 states;Frontiers in Molecular Biosciences;2022-11-08
5. Multiple Computational Approaches for Predicting Drug Interactions with Human Equilibrative Nucleoside Transporter 1;Drug Metabolism and Disposition;2021-05-12
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3