Inhibition of HIV-1 by non-nucleoside reverse transcriptase inhibitors via an induced fit mechanism—Importance of slow dissociation and relaxation rates for antiviral efficacy-Reference-Cited by-同舟云学术

Inhibition of HIV-1 by non-nucleoside reverse transcriptase inhibitors via an induced fit mechanism—Importance of slow dissociation and relaxation rates for antiviral efficacy

Published:2010-10 Issue:8 Volume:80 Page:1133-1140
ISSN:0006-2952
Container-title:Biochemical Pharmacology
language:en
Short-container-title:Biochemical Pharmacology

Author:

Elinder Malin,Selhorst Philippe,Vanham Guido,Öberg Bo,Vrang Lotta,Danielson U. Helena

Funder

Swedish International Development Cooperation Agency

Research Foundation–Flanders (FWO) Belgium

GE Healthcare Biosciences

Publisher

Elsevier BV

Subject

Pharmacology,Biochemistry

Reference20 articles.

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3. Development of non-nucleoside reverse transcriptase inhibitors for anti-HIV therapy;Sahlberg;Anti-Infective Agents in Medicinal Chemistry,2008

4. Concentrations of dapivirine in the rhesus macaque and rabbit following once daily intravaginal administration of a gel formulation of [14C]dapivirine for 7 days;Nuttall;Antimicrobial Agents and Chemotherapy,2008

5. Biosensor-based kinetic characterization of the interaction between HIV-1 reverse transcriptase and non-nucleoside inhibitors;Geitmann;Journal of Medicinal Chemistry,2006

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