Discovery of small molecule positive allosteric modulators of the secretin receptor-Reference-Cited by-同舟云学术

Discovery of small molecule positive allosteric modulators of the secretin receptor

Published:2021-03 Issue: Volume:185 Page:114451
ISSN:0006-2952
Container-title:Biochemical Pharmacology
language:en
Short-container-title:Biochemical Pharmacology

Author:

Dengler Daniela G.,Harikumar Kaleeckal G.,Pollari Sirkku,Sun Qing,Brown Brock T.,Shinoki-Iwaya Aki,Ardecky Robert,Miller Laurence J.,Sergienko Eduard A.

Funder

National Heart, Lung, and Blood Institute

National Institutes of Health

Publisher

Elsevier BV

Subject

Pharmacology,Biochemistry

Reference52 articles.

1. Structural basis for allosteric modulation of class B G Protein-Coupled Receptors;Wootten;Annu. Rev. Pharmacol. Toxicol.,2020

2. Allosteric modulators of class B G-protein-coupled receptors;Hoare;Curr. Neuropharmacol.,2007

3. The physiological roles of secretin and its receptor;Afroze;Ann. Transl. Med.,2013

4. Extending the structural view of class B GPCRs;de Graaf;Trends Biochem. Sci.,2017

5. Identification and Characterization of Dual-Acting Small Molecule Modulators targeting Secretin Receptors;Dengler;FASEB J.,2020

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