Determination of agonist dissociation constants in isolated vasculature: Equivalence of estimates obtained by the method of partial irreversible receptor inactivation and a novel application of the operational model of pharmacological agonism-Reference-Cited by-同舟云学术

Determination of agonist dissociation constants in isolated vasculature: Equivalence of estimates obtained by the method of partial irreversible receptor inactivation and a novel application of the operational model of pharmacological agonism

Published:1990 Issue:20 Volume:47 Page:1867-1874
ISSN:0024-3205
Container-title:Life Sciences
language:en
Short-container-title:Life Sciences

Author:

Christ George J.

Funder

U.S. Public Health Service

Publisher

Elsevier BV

Subject

General Pharmacology, Toxicology and Pharmaceutics,General Biochemistry, Genetics and Molecular Biology,General Medicine

Reference20 articles.

1. Beta-adrenergic receptors: biochemical mechanisms of physiological regulation

2. G proteins control diverse pathways of transmembrane signaling 1

3. An operational model of pharmacological agonism: the effect of E/[A] curve shape on agonist dissociation constant estimation

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