Use of endogenous cortisol 6β-hydroxylation clearance for phenotyping in vivo CYP3A activity in women after sequential administration of an oral contraceptive (OC) containing ethinylestradiol and levonorgestrel as weak CYP3A inhibitors-Reference-Cited by-同舟云学术

Use of endogenous cortisol 6β-hydroxylation clearance for phenotyping in vivo CYP3A activity in women after sequential administration of an oral contraceptive (OC) containing ethinylestradiol and levonorgestrel as weak CYP3A inhibitors

Published:2014-09 Issue: Volume:87 Page:137-144
ISSN:0039-128X
Container-title:Steroids
language:en
Short-container-title:Steroids

Author:

Shibasaki Hiromi,Kuroiwa Miyuki^ORCID,Uchikura Shinobu,Tsuboyama Sayuri,Yokokawa Akitomo,Kume Miyoko,Furuta Takashi

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Pharmacology,Endocrinology,Molecular Biology,Biochemistry

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4. Physiologically based pharmacokinetic model of mechanism-based inhibition of CYP3A by clarithromycin;Quinney;Drug Metab Dispos,2010

5. Mechanism of cytochrome P450-3A inhibition by ketoconazole;Greenblatt;J Pharm Pharmacol,2011

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