Drug–Target Association Kinetics in Drug Discovery
Author:
Funder
National Natural Science Foundation of China
Natural Science Foundation of Jiangsu Province
Publisher
Elsevier BV
Subject
Molecular Biology,Biochemistry
Reference88 articles.
1. Trial watch: phase II failures: 2008-2010;Arrowsmith;Nat. Rev. Drug Discov.,2011
2. An analysis of the attrition of drug candidates from four major pharmaceutical companies;Waring;Nat. Rev. Drug Discov.,2015
3. International Union of Pharmacology Committee on receptor nomenclature and drug classification. XXXVIII. Update on terms and symbols in quantitative pharmacology;Neubig;Pharmacol. Rev.,2003
4. The drug-target residence time model: a 10-year retrospective;Copeland;Nat. Rev. Drug Discov.,2016
5. The added value of assessing ligand-receptor binding kinetics in drug discovery;Guo;ACS Med. Chem. Lett.,2016
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