Molecular Diversity of Novel Amino Acid Based Dendrimers

Author:

Mulders Suzanne J.E.,Brouwer Arwin J.,Liskamp* Rob M.J.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference8 articles.

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2. a) Newkome, G.R.; Lin, X.; Weis, C.D. Tetrahedron Asymm. 1991, 2, 957; b) Uhrich, K.E.; Fréchet, J.M.J. J. Chem. Soc. Perkin Trans. 1 1992, 1623; c) Rao, C.; Tam, J.P. J. Am. Chem. Soc. 1994, 116, 6975; d) Shao, J.; Tam, J.P. J. Am. Chem. Soc. 1995, 117, 3893; e) Twymam, L.J.; Beezer, A.E.; Mitchell, J.C. Tetrahedron Lett. 1994, 35, 4423; f) Spetzler, J.C.; Tam, J.P. Int. J. Peptide Protein Res. 1995, 45, 78; g) Roy, R.; Park, W.K.C.; Wu, Q.; Wang, S-N. Tetrahedron Lett. 1995, 36, 4377; h) Zanini, D.; Park, W.K.C.; Roy, R. Tetrahedron Lett. 1995, 36, 7383; i) Dandliker, P.J.; Diederich, F.; Gross, M.; Knobler, C.B.; Louati, A.; Sanford, E.M. Angew. Chem. Int. Ed. Engl. 1994, 33, 1739; j) Dandliker, P.J.; Diederich, F.; Gisselbrecht, J.-P.; Louati, A.; Gross, M. Angew. Chem. Int. Ed. Engl. 1995, 34, 2725; k) Mattei, S.; Seiler, P.; Diederich, F.; Gramlich, V. Helv. Chim. Acta 1995, 78, 1904.

3. Synthesis of a novel amino acid based dendrimer

4. Reactifs de couplage peptidique I (1) - l'hexafluorophosphate de benzotriazolyl N-oxytrisdimethylamino phosphonium (B.O.P.)

5. For chiral dendrimers and dendrimers containing chiral groups see e.g. [2]a,c,e and a) Seebach, D.; Lapierre, J.-M.; Skobridis, K.; Greiveldinger, G. Angew. Chem. Int. Ed. Engl., 1994, 33, 440; b) Seebach, D.; Lapierre, J.-M.; Greiveldinger, G.; Skobridis, K. Helv. Chim. Acta, 1994, 77, 1673; c) Chow, H.-F.; Fok, L.F.; Mak, C.C. Tetrahedron Lett., 1994, 35, 3547; d) Kremers, J.A.; Meijer, E.W. J. Org. Chem., 1994, 59, 4262; e) Jansen, J.F.G.A.; Peerlings, H.W.I.; De Brabander van den Berg, E.M.M.; Meijer, E.W. Angew. Chem. Int. Ed. Engl. 1995, 34, 1206; f) Aoi, K.; Itoh, K.; Okada, M. Macromolecules, 1995, 28, 5391; g) Chang, H.T.; Chen, C.T.; Kondo, T.; Siuzdak, G.; Sharpless, K.B. Angew. Chem. Int. Ed. Engl. 1996, 35, 182. h) Mak, C.C.; Chow, H-F. Chem. Comm. 1996, 1185.

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