Interaction of bispyridinium compounds with the orthosteric binding site of human α7 and Torpedo californica nicotinic acetylcholine receptors (nAChRs)-Reference-Cited by-同舟云学术

Interaction of bispyridinium compounds with the orthosteric binding site of human α7 and Torpedo californica nicotinic acetylcholine receptors (nAChRs)

Published:2011-09 Issue:1 Volume:206 Page:100-104
ISSN:0378-4274
Container-title:Toxicology Letters
language:en
Short-container-title:Toxicology Letters

Author:

Niessen K.V.,Tattersall J.E.H.,Timperley C.M.,Bird M.,Green C.,Seeger T.,Thiermann H.,Worek F.

Publisher

Elsevier BV

Subject

Toxicology,General Medicine

Reference31 articles.

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3. Bis-azaaromatic quaternary ammonium analogues: ligands for α4β2 and α7 subtypes of neuronal nicotinic receptors;Ayers;Bioorg. Med. Chem. Lett.,2002

4. A rapid filtration assay for soluble receptors using polyethylenimine-treated filters;Bruns;Anal. Biochem.,1983

5. Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50 per cent inhibition (IC50) of an enzymatic reaction;Cheng;Biochem. Pharmacol.,1973

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