Rapid conversion of the ester prodrug abiraterone acetate results in intestinal supersaturation and enhanced absorption of abiraterone: In vitro, rat in situ and human in vivo studies-Reference-Cited by-同舟云学术

Rapid conversion of the ester prodrug abiraterone acetate results in intestinal supersaturation and enhanced absorption of abiraterone: In vitro, rat in situ and human in vivo studies

Published:2015-02 Issue: Volume:90 Page:1-7
ISSN:0939-6411
Container-title:European Journal of Pharmaceutics and Biopharmaceutics
language:en
Short-container-title:European Journal of Pharmaceutics and Biopharmaceutics

Author:

Stappaerts Jef,Geboers Sophie,Snoeys Jan,Brouwers Joachim,Tack Jan,Annaert Pieter,Augustijns Patrick

Funder

Scientific Research in Flanders (FWO)

‘Onderzoeksfonds’ of the KU Leuven in Belgium

Publisher

Elsevier BV

Subject

Pharmaceutical Science,General Medicine,Biotechnology

Reference12 articles.

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3. In vitro behavior of a phosphate ester prodrug of amprenavir in human intestinal fluids and in the Caco-2 system: illustration of intraluminal supersaturation;Brouwers;Int. J. Pharm.,2007

4. Stability of valacyclovir: implications for its oral bioavailability;Granero;Int. J. Pharm.,2006

5. Stability of cephalosporin prodrug esters in human intestinal juice: implications for oral bioavailability;Stoeckel;Antimicrob. Agents Chemother.,1998

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